{"product_id":"revvity-es-031-m400ua","title":"Revvity, ES-031-M400UA, Membrane Target Systems: Adrenergic α (human) membrane preparation, in CHO-K1 cells. 400 Units.","description":"\u003cp\u003eOverview\u003cbr\u003e\nMembrane Target Systems are quality assured frozen membranes from cells that express Adrenergic alpha 2B (human) recombinant or endogenous receptors.\u003cbr\u003e\nWe submit every batch of receptor to stringent quality controltesting that includes saturation radioligand binding assay todetermine receptor concentration (Bmax) and affinity (Kd).Competition binding assays are performed determine affinity (Ki)against known reference agonists and antagonists. GTPgS data isalso provided for some of our Gi coupled receptors.\u003cbr\u003e\nMembranes are carefully prepared and ready for a variety of HTSapplications, including radioligand binding (using either proximitymethods, such as FlashPlate, or classical filtrationmethods).\u003cbr\u003e\nProducts are packaged as frozen crude membrane preparations. Oneassay unit is defined as micrograms of protein, defined bycompetition binding assay (filtration). A complete productdescription and recommended protocol are included on the ProductInformation Sheet.\u003cbr\u003e\nSome of our receptors may be restricted for sale in specifiedcountries. Please inquire. Concentration-5 µg\/µL protein\u003cbr\u003e\nVolume-400.0 µL\u003cbr\u003e\nµg protein\/unit-5 µg protein \/ unit\u003c\/p\u003e\n\n\u003cp\u003eApplication-Drug Discovery \u0026amp; Development\u003cbr\u003e\nBrand-Membrane Target Systems\u003cbr\u003e\nBuffer\/Solvent-50 mM Tris-HCL (pH 7.4), 0.5mM EDTA, 10mM MgCl2, 10% sucrose\u003cbr\u003e\nG-Alpha Natural Receptor-G i \/G o\u003cbr\u003e\nHost Cell Line-CHO-K1\u003cbr\u003e\nHost Species-Human\u003cbr\u003e\nProduct Group-Membrane Preparation\u003cbr\u003e\nReceptor-Adrenergic\u003cbr\u003e\nSecond Messenger Release-GTP exchange\u003cbr\u003e\nShipping Conditions-Shipped in Dry Ice\u003cbr\u003e\nTarget Class-GPCR\u003cbr\u003e\nTherapeutic Area-Cardiovascular Diabetes Gastrointestinal Inflammation Metabolic\u003cbr\u003e\nUnit Size-400 units\u003cbr\u003e\nValidation-Binding GTPγS\u003c\/p\u003e","brand":"Revvity","offers":[{"title":"Default Title","offer_id":46774514319529,"sku":"ES-031-M400UA","price":0.99,"currency_code":"USD","in_stock":true}],"url":"https:\/\/iright.com\/products\/revvity-es-031-m400ua","provider":"Iright","version":"1.0","type":"link"}