{"product_id":"revvity-es-621-m400ua","title":"Revvity, ES-621-M400UA, Membrane Target Systems: Melatonin MT2 (human) membrane preparation, in CHO-K1 cells. 400 Units.","description":"\u003cp\u003eOverview\u003cbr\u003e\nMembrane Target Systems are quality assured frozen membranes from cells that express Melatonin MT2 (human) recombinant or endogenous receptors. We submit every batch of receptor to stringent quality control testing that includes saturation radioligand binding assay to determine receptor concentration (Bmax) and affinity (Kd). Competition binding assays are performed determine affinity (Ki) against known reference agonists and antagonists. GTPgS data is also provided for some of our Gi coupled receptors.\u003cbr\u003e\nMembranes are carefully prepared and ready for a variety of HTS applications, including radioligand binding (using either proximity methods, such as FlashPlate, or classical filtration methods).\u003cbr\u003e\nProducts are packaged as frozen crude membrane preparations. One assay unit is defined as micrograms of protein, defined by competition binding assay (filtration). A complete product description and recommended protocol are included on the Product Information Sheet (see Certificate of Analysis). Concentration-2.5 µg\/µL protein\u003cbr\u003e\nVolume-400.0 µL\u003cbr\u003e\nµg protein\/unit-2.5 µg protein \/ unit\u003cbr\u003e\nApplication-Drug Discovery \u0026amp; Development\u003cbr\u003e\nBrand-Membrane Target Systems\u003cbr\u003e\nBuffer\/Solvent-50 mM Tris-HCL (pH 7.4), 0.5mM EDTA, 10mM MgCl2, 10% sucrose\u003cbr\u003e\nG-Alpha Natural Receptor-G i \/G o\u003cbr\u003e\nHost Cell Line-CHO-K1\u003cbr\u003e\nHost Species-Human\u003cbr\u003e\nProduct Group-Membrane Preparation\u003cbr\u003e\nReceptor-Melatonin\u003cbr\u003e\nShipping Conditions-Shipped in Dry Ice\u003cbr\u003e\nTarget Class-GPCR\u003cbr\u003e\nTherapeutic Area-Cardiovascular Central Nervous System\u003cbr\u003e\nUnit Size-400 units\u003cbr\u003e\nValidation-Binding\u003c\/p\u003e","brand":"Revvity","offers":[{"title":"Default Title","offer_id":46775346856105,"sku":"ES-621-M400UA","price":0.99,"currency_code":"USD","in_stock":true}],"url":"https:\/\/iright.com\/products\/revvity-es-621-m400ua","provider":"Iright","version":"1.0","type":"link"}