{"product_id":"revvity-nex174100uc","title":"Revvity, NEX174100UC, iodo-(±)-Cyanopindolol, [ I], 100µCi (3.7MBq)","description":"\u003cp\u003eOverview\u003cbr\u003e\n100 µCi Quantities of iodo-(±)-Cyanopindolol, [125I], are available for your research.\u003cbr\u003e\nWe offer radioligands and radiolabeled biomolecules to use as tracers, for radioimmunoassays (RIAs), for autoradiographic visualization, or for performing saturation and competition radioligand binding assays to determine receptor expression levels (Bmax), dissociation constants (Kd), association and dissociation rates (kon and koff), and inhibitor constants (Ki) for a variety of receptors. We develop our radioligands to the highest specific activity possible and provide high purity resulting in low non-specific binding products. Each of our ultra-pure radiolabeled compounds is fully characterized for pharmacological action and validated in binding assays.\u003cbr\u003e\nRadiochemicals remain the most sensitive method for probing binding biology; yielding unprecedented sensitivity gives results that technicians and scientists can trust. For over 50 years, Revvity has been a leading supplier of New England Nuclear (NEN) radiochemicals, liquid scintillation cocktails, vials and nuclear counting detection instruments.\u003cbr\u003e\nReferences for NEX174:\u003c\/p\u003e\n\n\u003cp\u003eFlügge, G., Ahrens, O. \u0026amp; Fuchs, E. (1997) β-Adrenoceptors in the Tree Shrew Brain. II. Time-Dependent Effects of Chronic Psychosocial Stress on [125I]Iodocyanopindolol Binding Sites, Cell Mol Neurobiol 17: 417-432.\u003cbr\u003e\nPei, G., Samama, P., Lohse, M., Wang, M., Codina, J., Lefkowitz, R.J. (1994), A constitutively active mutant beta 2-adrenergic receptor is constitutively desensitized and phosphorylated, PNAS, 91 (7): 2699-2702. Molecular Weight-411\u003cbr\u003e\nCAS Number-85124-14-7\u003cbr\u003e\nApplication-Drug Discovery \u0026amp; Development\u003cbr\u003e\nBrand-NEN Radiochemicals\u003cbr\u003e\nBuffer\/Solvent-1 propanaol : water : phenol (~50:50:1 2)\u003cbr\u003e\nDetection Modality-Radiometric\u003cbr\u003e\nFresh Lot Days-First Monday of each month\u003cbr\u003e\nLabel Position-Nominally Labeled\u003cbr\u003e\nMolecular Formula-C16H20IN3O2\u003cbr\u003e\nPackaging-NENSure vial\u003cbr\u003e\nRadioisotope-125 I\u003cbr\u003e\nReceptor-Adrenoceptors\u003cbr\u003e\nShipping Information-Shipped on Dry Ice\u003cbr\u003e\nShipping Conditions-Shipped in Dry Ice\u003cbr\u003e\nSpecial Ordering Information-This is a radioactive product - shipping address must have a license to receive radioactive materials.\u003cbr\u003e\nStorage Conditions-4°C\u003cbr\u003e\nTherapeutic Area-Cardiovascular CNS \u0026amp; Neurologic Metabolic Disorders\u003cbr\u003e\nUnit Size-100 µCi\u003c\/p\u003e","brand":"Revvity","offers":[{"title":"Default Title","offer_id":46775200252073,"sku":"NEX174100UC","price":0.99,"currency_code":"USD","in_stock":true}],"url":"https:\/\/iright.com\/products\/revvity-nex174100uc","provider":"Iright","version":"1.0","type":"link"}