Abcam, ab120923, Leelamine, Pyruvate dehydrogenase kinase (PDK) inhibitor

Size: 10mg / 50mg
MW 285.47 g/mol, Purity >98%. Pyruvate dehydrogenase kinase (PDK) inhibitor (IC 50 = 9.5 μM). It has weak affinity for human CB 1 and CB 2 receptors, exhibiting 20% displacement of [3H]-CP55940 at a concentration of 10 μM.
Key facts
CAS number:1446-61-3,
Purity:>98%,
Form:LiquidSee storage information,
Molecular weight:285.47 g/mol,
Molecular formula:C20H31N,
Nature:Synthetic,
Biological description:Pyruvate dehydrogenase kinase (PDK) inhibitor (IC50 = 9.5 μM). It has weak affinity for human CB1 and CB2 receptors, exhibiting 20% displacement of [3H]-CP55940 at a concentration of 10 μM.,
Isomeric smiles:CC(C)C(C=C1)=CC2=C1[C@]3(C)[C@](CC2)([H])[C@@](CN)(C)CCC3,
IUPAC Name:(1R,4aS,10aR)-1,2,3,4,4a,9,10,10a-Octahydro-1,4a-dimethyl-7-(1-methylethyl)-1-phenanthrenemethanamine

Properties and Storage Information:
Shipped at conditions-Ambient - Can Ship with Ice, Appropriate short-term storage conditions-Ambient, Appropriate long-term storage conditions-Ambient