Abcam, ab120317, NNC 05-2090, GABA uptake inhibitor

Size: 10mg / 50mg
MW 451 Da, Purity >99%. GABA uptake inhibitor, selective for the BGT-1 transporter (K i values are 1.4 (BGT-1), 19 (GAT-1), 41 (GAT-2) and 15 μM (GAT-3)). Also active at α 1 - and D 2 -receptors (IC 50 values are 266 and 1632 nM, respectively). Anticonvulsant in vivo .
Key facts
CAS number:184845-43-0,
Purity:>99%,
Form:SolidSee storage information,
Molecular weight:451 Da,
Molecular formula:C27H31ClN2O2,
PubChem:18782760,
Nature:Synthetic,
Solubility:Soluble in DMSO to 100 mM,
Biochemical name:1-[3-(9H-Carbazol-9-YL)propyl]-4-(2-methoxyphenyl)-4-piperidinol hydrochloride,
Biological description:GABA uptake inhibitor, selective for the BGT-1 transporter (Ki values are 1.4 (BGT-1), 19 (GAT-1), 41 (GAT-2) and 15 μM (GAT-3)). Also active at α1- and D2-receptors (IC50 values are 266 and 1632 nM, respectively). Anticonvulsant in vivo.,
Canonical smiles:COC1=CC=CC=C1C2(CCN(CC2)CCCN3C4=CC=CC=C4C5=CC=CC=C53)O.Cl,
InChi:InChI=1S/C27H30N2O2.ClH/c1-31-26-14-7-4-11-23(26)27(30)15-19-28(20-16-27)17-8-18-29-24-12-5-2-9-21(24)22-10-3-6-13-25(22)29;/h2-7,9-14,30H,8,15-20H2,1H3;1H,
InChiKey:WDFXPKKFSNMGOO-UHFFFAOYSA-N,
IUPAC Name:1-(3-carbazol-9-ylpropyl)-4-(2-methoxyphenyl)piperidin-4-ol;hydrochloride

Properties and Storage Information:
Shipped at conditions-Ambient - Can Ship with Ice, Appropriate short-term storage conditions-Ambient, Appropriate long-term storage conditions-Ambient, Storage information-Store under desiccating conditions, The product can be stored for up to 12 months