Abcam, ab120042, SR95531 (Gabazine), GABAA antagonist

Size: 10mg / 50mg
SR95531 (Gabazine) is a selective, competitive GABAA receptor antagonist. Allosteric inhibitor of channel opening of the GABAA receptor. Displaces [3H]-GABA from rat brain membranes with a Ki of 150 nM. MW 368.23. - Available in different sizes to fit your experimental needs
Key facts
CAS number:104104-50-9,
Purity:>98%,
Form:SolidSee storage information,
Molecular weight:368.23 Da,
Molecular formula:C15H18BrN3O3,
PubChem:107895,
Nature:Synthetic,
Biochemical name:1(6H)-Pyridazinebutanoic acid, 6-imino-3-(4-methoxyphenyl)-, monohydrobromide,
Biological description:Selective, competitive GABAA receptor antagonist. Allosteric inhibitor of channel opening of the GABAA receptor. Displaces [3H]-GABA from rat brain membranes with a Ki of 150 nM. Soluble in 1 ml water to give specified mM/ml concentration.,
Canonical smiles:COC1=CC=C(C=C1)C2=NN(C(=N)C=C2)CCCC(=O)O.Br,
InChi:InChI=1S/C15H17N3O3.BrH/c1-21-12-6-4-11(5-7-12)13-8-9-14(16)18(17-13)10-2-3-15(19)20;/h4-9,16H,2-3,10H2,1H3,(H,19,20);1H,
InChiKey:GFZHNFOGCMEYTA-UHFFFAOYSA-N,
IUPAC Name:4-[6-imino-3-(4-methoxyphenyl)pyridazin-1-yl]butanoic acid;hydrobromide

Product details:
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Properties and Storage Information:
Shipped at conditions-Ambient - Can Ship with Ice, Appropriate short-term storage conditions-+4°C, Appropriate long-term storage conditions-+4°C, Storage information-Store under desiccating conditions, The product can be stored for up to 12 months