Abcam, ab120523, GR 127935 hydrochloride, 5-HT1B/1D receptor antagonist

Size: 10mg / 50mg
MW 534.06 g/mol, Purity >97%. Potent and selective 5-HT 1B/1D receptor antagonist (pK i = 8.5 for both 5-HT 1D in rat and 5-HT 1D in guinea pig). 100-fold selectivity over 5-HT 1A , 5-HT 1E , and 5-HT 2C . Displays centrally mediated effects upon systemic administration.
Key facts
CAS number:148642-42-6,
Purity:>97%,
Form:SolidSee storage information,
Molecular weight:534.06 g/mol,
Nature:Synthetic,
Solubility:Soluble in water to 25 mM,
Biological description:Potent and selective 5-HT1B/1D receptor antagonist (pKi = 8.5 for both 5-HT1D in rat and 5-HT1D in guinea pig). 100-fold selectivity over 5-HT1A, 5-HT1E, and 5-HT2C. Displays centrally mediated effects upon systemic administration.,
IUPAC Name:N-[4-Methoxy-3-(4-methyl-1-piperazinyl)phenyl]-2'-methyl-4'-(5-methyl-1,2,4-oxadiazol-3-yl)-1,1'-biphenyl-4-carboxamide hydrochloride

Properties and Storage Information:
Shipped at conditions-Ambient - Can Ship with Ice, Appropriate short-term storage conditions-+4°C, Appropriate long-term storage conditions-+4°C, Storage information-Store under desiccating conditions, The product can be stored for up to 12 months