Abcam, ab141106, YIL781 hydrochloride, Ghrelin receptor antagonist

Size: 10mg / 50mg
MW 445.96 g/mol, Purity >99%. Ghrelin receptor (GHS-R1a) antagonist (K i = 17 nM). Competitive antagonist activity in vitro (pK B = 7.54). Displays no affinity for the motilin receptor (K i = 6 μM).
Key facts
CAS number:875258-85-8,
Purity:>99%,
Form:SolidSee storage information,
Molecular weight:445.96 g/mol,
Molecular formula:C24H28FN3O2.HCl,
Nature:Synthetic,
Solubility:Soluble in DMSO to 100 mMSoluble in ethanol to 100 mM,
Biological description:Ghrelin receptor (GHS-R1a) antagonist (Ki = 17 nM). Competitive antagonist activity in vitro (pKB = 7.54). Displays no affinity for the motilin receptor (Ki = 6 μM).,
Isomeric smiles:CL.CC(C)N4CCC[C@H](CN3C(C)=NC2CCC(OC1CCC(F)CC1)CC2C3=O)C4,
InChi:InChI=1S/C24H28FN3O2.ClH/c1-16(2)27-12-4-5-18(14-27)15-28-17(3)26-23-11-10-21(13-22(23)24(28)29)30-20-8-6-19(25)7-9-20;/h6-11,13,16,18H,4-5,12,14-15H2,1-3H3;1H/t18-;/m0./s1,
InChiKey:QQGRMONBDBMLSP-FERBBOLQSA-N,
IUPAC Name:6-(4-Fluorophenoxy)-2-methyl-3-[[(3S)-1-(1-methylethyl)-3-piperidinyl]methyl]-4(3H)-quinazolinone hydrochloride

Properties and Storage Information:
Shipped at conditions-Ambient - Can Ship with Ice, Appropriate short-term storage conditions-Ambient, Appropriate long-term storage conditions-Ambient, Storage information-Store under desiccating conditions, The product can be stored for up to 12 months